Analysis of argyrin B binding at constitutive and immunoproteasome active sites using molecular modelling and kinetic assays

Conference poster

Allardyce, D., Bell, C. and Loizidou, E. 2017. Analysis of argyrin B binding at constitutive and immunoproteasome active sites using molecular modelling and kinetic assays. Computational Advances in Drug Discovery (Structure Based Drug Design). Lausanne, Switzerland 05 - 08 Sep 2017
TypeConference poster
TitleAnalysis of argyrin B binding at constitutive and immunoproteasome active sites using molecular modelling and kinetic assays
AuthorsAllardyce, D., Bell, C. and Loizidou, E.
ConferenceComputational Advances in Drug Discovery (Structure Based Drug Design)
Publication dates
Print03 Sep 2017
Publication process dates
Deposited23 Feb 2018
Accepted30 Jun 2017
Output statusPublished
LanguageEnglish
Permalink -

https://repository.mdx.ac.uk/item/87798

Log in to edit

Restricted files

First submitted version

  • 60
    total views
  • 0
    total downloads
  • 0
    views this month
  • 0
    downloads this month

Export as

Related outputs

Identification of a new class of proteasome inhibitors based on a naphthyl-azotricyclic-urea-phenyl scaffold
Allardyce, D., Adu Mantey, P., Szalecka, M., Nkwo, R. and Loizidou, E. 2023. Identification of a new class of proteasome inhibitors based on a naphthyl-azotricyclic-urea-phenyl scaffold. RSC Medicinal Chemistry. 14 (3), pp. 573-582. https://doi.org/10.1039/D2MD00404F
Intentionality for inclusivity - the journey at Middlesex University
Roberts, H., Punev, I., Allardyce, D., Kyprianou, A., Appiah, S., Megeney, A., Calin, A., Gallacher, D. and Mill, R. 2022. Intentionality for inclusivity - the journey at Middlesex University. McGraw Hill.
Argyrin B a non-competitive inhibitor of the human immunoproteasome exhibiting preference for β1i
Allardyce, D., Bell, C. and Loizidou, E. 2019. Argyrin B a non-competitive inhibitor of the human immunoproteasome exhibiting preference for β1i. Chemical Biology and Drug Design. 94 (2), pp. 1556-1567. https://doi.org/10.1111/cbdd.13539
Biochemical and computational studies towards selective inhibition of the immunoproteasome
Allardyce, D. 2018. Biochemical and computational studies towards selective inhibition of the immunoproteasome. Masters thesis Middlesex University Natural Sciences